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USMLE - Autonomic Drugs Part 1

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This deck most postganglionic fibers release norepinephrine; however, there are exceptions.

Sympathetic Nervous System organs innervated by cholinergic fibers?

Sweat glands and Adrenal Medulla

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Key Terms

Term
Definition

Sympathetic Nervous System organs innervated by cholinergic fibers?

Sweat glands and Adrenal Medulla

Botulinum Toxin

Prevents release of ACh at all cholinergic terminals

Nicotinic ACh receptors

Description

Location?

Ligand gated Na/K channel

Autonomic ganglia and NMJ

α1

System

Kind of receptor?

Class

Function

Sympathetic

GPCR

q

Vascular SM contraction, Pupillary dilator muscle contraction (mydriasis), Intestinal and Bladder Sphincter mu...

α2

System

Kind of receptor?

Class

Function

Sympathetic

GPCR

i

↓ sympathetic outflow, ↓ insulin release, ↓ lipolysis, ↑ platelet aggregation

β1

System

Kind of receptor?

Class

Function

Sympathetic

GPCR

s

↑ HR, contractility, rennin release, lipolysis

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TermDefinition

Sympathetic Nervous System organs innervated by cholinergic fibers?

Sweat glands and Adrenal Medulla

Botulinum Toxin

Prevents release of ACh at all cholinergic terminals

Nicotinic ACh receptors

Description

Location?

Ligand gated Na/K channel

Autonomic ganglia and NMJ

α1

System

Kind of receptor?

Class

Function

Sympathetic

GPCR

q

Vascular SM contraction, Pupillary dilator muscle contraction (mydriasis), Intestinal and Bladder Sphincter muscle contraction

α2

System

Kind of receptor?

Class

Function

Sympathetic

GPCR

i

↓ sympathetic outflow, ↓ insulin release, ↓ lipolysis, ↑ platelet aggregation

β1

System

Kind of receptor?

Class

Function

Sympathetic

GPCR

s

↑ HR, contractility, rennin release, lipolysis

β2

System

Kind of receptor?

Class

Function

Sympathetic

GPCR

s

Vasodilation, Bronchodilation, ↓ Uterine Tone (tocolysis)

↑ HR, contractility, lipolysis, insulin release

Ciliary Muscle Relaxation and ↑ Aqueous Humor production

M1

System

Kind of receptor?

Class

Function

Parasympathetic

GPCR

q

CNS, Enteric Nervous System

M2

System

Kind of receptor?

Class

Function

Parasympathetic

GPCR

i

↓ HR and atrai contractility

M3

System

Kind of receptor?

Class

Function

Parasympathetic

q

GPCR

Exocrine gland secretion, gut peristalsis, bladder contraction, Bronchoconstriction, Pupillary sphincter muscle contraction (Miosis), Ciliary muscle contraction (accommodation)

D1

Kind of receptor?

Class

Function

GPCR

s

Relaxes renal vascular smooth muscle

D2

Kind of receptor?

Class

Function

GPCR

i

Modulates transmitter release, esp in brain

H1

Kind of receptor?

Class

Function

GPCR

q

Nasal and Bronchial mucus production, contraction of bronchioles, pruritus, pain

H2

Kind of receptor?

Class

Function

GPCR

s

Gastric Acid Secretion

V1

Kind of receptor

Class

Function

GPCR

q

Vascular smooth muscle contraction

V2

Kind of receptor

Class

Function

GPCR

s

↑ water permeability and reabsorption in collecting tubule of kidneys

Autonomic Receptor Mnemonic

QISS and QIQ until you're SIQ of SQS

α1, α2, β1, β2

M1, M2, M3

D1, D2

H1, H2

V1, V2

Autonomic drugs that use IP3/DAG

“HAVe 1 M&M”

H1, α1, V1, M1, M3

Autonomic drugs that ↓ cAMP

“MAD2”

M2, α2, D2

Autonomic drugs that ↑ cAMP

Gs

“Bill Bob Doesn’t Have Value”

β1, β2, D1, H2, V2

Hemicholinium

Blocks re-uptake of choline at ACh nerve terminal

Vesamicol

Blocks ACh packaging into vesicles

Metyrosine

Inhibits conversion of Tyrosine to DOPA

Reserpine

Inhibits packaging of DA into vesicles

May be turned into NE in vesicle

Guanethidine

Inhibits release of NE